Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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121
Tocris Bioscience™ MONNA, >98%
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CAS: 1572936-83-4 Molecular Formula: C18H14N2O5
| CAS | 1572936-83-4 |
|---|---|
| Molecular Formula | C18H14N2O5 |
122
Tocris Bioscience™ SCH 336
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Highly potent and selective CB2 inverse agonist
| CAS | 447459-51-0 |
|---|---|
| Chemical Name or Material | N-[(1S)-1-[4-[[4-Methoxy-2-[(4-methoxyphenyl)sulfonyl]phenyl]sulfonyl]phenyl]ethyl]methanesulfonamide |
| Recommended Storage | Store at Room Temperature |
| Molecular Formula | C23H25NO8S3 |
| Formula Weight | Observed MW: 539.64 |
| Assay Percent Range | >98% |
123
Tocris Bioscience™ Ambrisentan
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Selective ETA antagonist
124
Tocris Bioscience™ Ex 26
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Potent and selective S1P1 receptor antagonist
| CAS | 1233332-37-0 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Color | White |
| Solubility | Soluble to 100mM in DMSO and to 100mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | 1-[[[5'-[[1-(4-Chloro-3-methylphenyl)ethyl]amino]-2'-fluoro-3,5-dimethyl[1,1'-biphenyl]-4-yl]carbonyl]amino]-cyclopropanecarboxylic acid |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C28H28ClFN2O3 |
| Formula Weight | 494.98 |
125
Tocris Bioscience™ JZP 361, >99%
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Potent and selective reversible MAGL inhibitor
| CAS | 1680193-80-9 |
|---|---|
| Solubility | Soluble to 100mM in DMSO and to 20mM in ethanol |
| Purity | >99% |
| Chemical Name or Material | [4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl](1H-1,2,4- |
| Recommended Storage | Store at 4deg;C |
| Formula Weight | 405.88 |
126
Tocris Bioscience™ Ritonavir
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HIV-1 and HIV-2 protease inhibitor
127
Tocris Bioscience™ Imatinib mesylate
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Potent and selective v-Abl tyrosine kinase inhibitor; also inhibits PDGFR and c-kit
128
Tocris Bioscience™ H2DCFDA, >97%
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CAS: 4091-99-0 Molecular Formula: C24H16Cl2O7
| CAS | 4091-99-0 |
|---|---|
| Molecular Formula | C24H16Cl2O7 |
129
Tocris Bioscience™ Perifosine
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PKB/Akt inhibitor; also modulates Kv2.1 current
| CAS | 157716-52-4 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Color | White |
| Solubility | Soluble to 100mM in water and to 100mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | Perifosine |
| Recommended Storage | Store at -20°C |
| Synonym | Octadecyl-(1,1-dimethyl-4-piperidylio) phosphate |
| Molecular Formula | C25H52NO4P |
| Formula Weight | 461.66 |
130
Tocris Bioscience™ OB 24 hydrochloride
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Potent and selective heme oxygenase 1 (HO-1) inhibitor
| CAS | 939825-12-4 |
|---|---|
| Chemical Name or Material | 1-[[2-[2-(4-Bromophenyl)ethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazole hydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C15H17BrN2O2.HCl |
| Formula Weight | Observed MW: 373.67 |
| Assay Percent Range | >98% |
131
Tocris Bioscience™ MS 21570
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GPR171 antagonist
| CAS | 65373-29-7 |
|---|---|
| Chemical Name or Material | N-Methyl-5-[(phenylmethyl)thio]-1,3,4-thiazadiazol-2-amine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C10H11N3S2 |
| Formula Weight | Observed MW: 237.34 |
| Assay Percent Range | >98% |
132
Tocris Bioscience™ Thalidomide 4'-oxyacetamide-alkylC4-azide
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Azide-functionalized Thalidomide; click cereblon ligand for PROTACs
133
Tocris Bioscience™ ST 034307
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CAS: 133406-29-8 Molecular Formula: C10H4Cl4O2
| CAS | 133406-29-8 |
|---|---|
| Molecular Formula | C10H4Cl4O2 |
134
Tocris Bioscience™ KYP 2047
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High affinity prolyl oligopeptidase inhibitor (Ki = 0.023 nM); anti-angiogenic, neuroprotective and brain penetrant
| CAS | 796874-99-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (2S)-1-[[(2S)-1-(1-Oxo-4-phenylbutyl)-2-pyrrolidinyl]carbonyl]-2-pyrrolidinecarbonitrile |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H25N3O2 |
| Formula Weight | 339.44 |
135
Tocris Bioscience™ GSK 2239633A
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Potent CCR4 antagonist
| CAS | 1240516-71-5 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[[3-[[3-[[(5-Chloro-2-thienyl)sulfonyl]amino]-4-methoxy-1H-indazol-1-yl]methyl]phenyl]methyl]-2-hydroxy-2-methylpropanamide |
| Molecular Formula | C24H25ClN4O5S2 |